SCHEMBL7984133

SCHEMBL7984133

Cc1ncc(-c2cccc(N=C(N)N)c2)n1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 6/20 0.47
HTR3B O95264 6/20 0.47
HTR3A P46098 6/20 0.47
HTR3D Q70Z44 6/20 0.47
HTR3C Q8WXA8 6/20 0.47
SLC22A2 O15244 1/20 0.44
SLC22A1 O15245 1/20 0.44
SLC22A3 O75751 1/20 0.44
PLAU P00749 1/20 0.44
PRMT5 O14744 1/20 0.41
WDR77 Q9BQA1 1/20 0.41
KDM1A O60341 1/20 0.41
TAAR1 Q96RJ0 1/20 0.40
ADRA2A P08913 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
USP2 O75604 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7122972 0.99 HTR3E (0.46) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7125602 0.78 TTK (0.39) PRMT5WDR77DYRK1AGSK3BWNT1
SCHEMBL6754326 0.76 MAP4K4 (0.49) PRMT5WDR77CYP1A2CYP3A4CYP2D6
SCHEMBL6756716 0.76 FYN (0.54) DYRK1AGSK3B
SCHEMBL7122138 0.75 NPFFR1 (0.39) DYRK1AGSK3BWNT1
SCHEMBL7117412 0.74 DYRK1A (0.39) MAPTDYRK1AGSK3BWNT1
SCHEMBL7128738 0.73 MAPT (0.51) PRMT5WDR77CYP1A2CYP3A4CYP2D6
SCHEMBL7984129 0.73 FGFR3 (0.42) DYRK1AGSK3BWNT1
SCHEMBL7121296 0.73 CYP1A2 (0.50) CYP1A2DYRK1AGSK3BWNT1
Hydrochloric Acid SCHEMBL7123999 0.72 FGFR3 (0.41) DYRK1AGSK3BWNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001087845-A2 N-CONTAINING HETEROCYCLIC COMPOUNDS AND THEIR USE AS 5-HT ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-22 WO disclosed