Bromide

Bromide

SCHEMBL7984185

Br.Nc1ccc2c(c1N)CCN(Cc1cccc(C(F)(F)F)c1)C2

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 known ✓ P20309 1/20 0.40
SIGMAR1 known ✓ Q99720 1/20 0.40
ALDH1A1 P00352 2/20 0.51
GAA P10253 2/20 0.51
KDM4E B2RXH2 1/20 0.51
BRS3 P32247 1/20 0.48
LMNA P02545 2/20 0.47
ADORA1 P30542 1/20 0.46
DRD2 P14416 1/20 0.45
DRD3 P35462 1/20 0.45
KCNH2 Q12809 1/20 0.45
TACR1 P25103 2/20 0.42
FAAH O00519 1/20 0.40
PARP1 P09874 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
OPRL1 P41146 2/20 0.39
ACACB O00763 1/20 0.38
KDR P35968 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL7981194 0.86 KDM4E (0.47) ALDH1A1GAAKDM4EDRD2DRD3
SCHEMBL7987036 0.81 KDM4E (0.50) ALDH1A1GAAKDM4EBRS3LMNA
SCHEMBL1854844 0.80 KDM4E (0.54) ALDH1A1GAAKDM4EBRS3LMNA
SCHEMBL6974043 0.80 KDM4E (0.54) ALDH1A1GAAKDM4EBRS3LMNA
SCHEMBL7984647 0.75 KDM4E (0.48) ALDH1A1GAAKDM4EDRD2DRD3
SCHEMBL4985989 0.74 KDM4E (0.50) ALDH1A1GAAKDM4EBRS3LMNA
SCHEMBL2439744 0.74 KDM4E (0.62) ALDH1A1GAAKDM4EBRS3LMNA
SCHEMBL1854687 0.73 KDM4E (0.54) ALDH1A1GAAKDM4EBRS3LMNA
SCHEMBL697853 0.72 KDM4E (0.53) ALDH1A1GAAKDM4EBRS3LMNA
SCHEMBL7983703 0.72 BRS3 (0.45) ALDH1A1GAAKDM4EBRS3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6197771-B1 NERVOUS SYSTEM DISORDERS; ANTIISCHEMIC AGENTS; ALZHEIMER'SDISEASE; PARKINSON'S DISEASE; HUNTINGTON'S DISEASE WARNER-LAMBERT COMPANY 2001-03-06 US claimed