SCHEMBL6974043

SCHEMBL6974043

Nc1ccc2c(c1)CCN(Cc1cccc(C(F)(F)F)c1)C2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.54
ALDH1A1 P00352 1/20 0.54
GAA P10253 1/20 0.54
DRD3 P35462 2/20 0.50
LMNA P02545 1/20 0.50
DRD2 P14416 1/20 0.50
KCNH2 Q12809 1/20 0.50
ACACB O00763 1/20 0.47
BRS3 P32247 1/20 0.46
HTR1A P08908 2/20 0.45
TACR1 P25103 2/20 0.44
SIGMAR1 Q99720 3/20 0.44
ADORA1 P30542 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
DRD4 P21917 2/20 0.43
HTR2B P41595 2/20 0.43
TMEM97 Q5BJF2 2/20 0.43
MAOB P27338 2/20 0.43
CHRM2 P08172 1/20 0.43
CHRM3 P20309 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6972571 0.84 DRD2 (0.55) KDM4EALDH1A1DRD3DRD2KCNH2
SCHEMBL6973388 0.82 TMEM97 (0.60) DRD3DRD2KCNH2HTR1ASIGMAR1
SCHEMBL29438588 0.81 OPRM1 (0.44) KDM4EALDH1A1GAADRD3LMNA
SCHEMBL6972464 0.81 SIGMAR1 (0.52) KDM4EALDH1A1GAADRD3DRD2
SCHEMBL6974431 0.81 DRD4 (0.48) KDM4EALDH1A1GAADRD3HTR1A
SCHEMBL6965841 0.81 CA9 (0.50) KDM4EALDH1A1DRD3HTR1ASIGMAR1
Bromide SCHEMBL7984185 0.80 ALDH1A1 (0.51) KDM4EALDH1A1GAADRD3LMNA
SCHEMBL697853 0.80 KDM4E (0.53) KDM4EALDH1A1GAADRD3LMNA
SCHEMBL6966787 0.78 KMT2A (0.60) BRS3SIGMAR1
SCHEMBL6971135 0.78 SIGMAR1 (0.66) KDM4EALDH1A1DRD3DRD2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832069-B1 BIPHENYL-2-CARBOXYLIC ACID-TETRAHYDRO-ISOQUINOLIN-6-YL AMIDE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS INHIBITORS OF MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN AND/OR APOLIPOPROTEIN B (Apo B) SECRETION PFIZER (US) 2003-03-05 EP disclosed
EP-1181954-A2 Biphenyl-2-carboxylic acid-tetrahydro-isoquinolin-6-yl amide derivatives, their preparation and use as inhibitors of microsomal triglyceride transfer protein and/or apolipoprotein B (ApoB) secretion PFIZER INC. (US) 2002-02-27 EP disclosed