SCHEMBL7984420

SCHEMBL7984420

Cc1ncc(-c2cccc([AsH]c3nccc4c(-c5ccc(F)cc5)cccc34)c2)n1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 7/20 0.38
GSK3B P49841 3/20 0.38
WNT1 P04628 2/20 0.36
TTK P33981 3/20 0.36
CLK2 P49760 2/20 0.36
CLK3 P49761 2/20 0.36
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
GAA P10253 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
MAPK1 P28482 2/20 0.33
ATP1A1 P05023 1/20 0.33
ATP1B1 P05026 1/20 0.33
ATP1A3 P13637 1/20 0.33
ATP1B2 P14415 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7125034 0.78 RIPK2 (0.42) DYRK1AGSK3BWNT1TTKCLK2
SCHEMBL14077014 0.69 GAA (0.54) DYRK1AGSK3BKDM4EALDH1A1GAA
SCHEMBL18448007 0.67 WNT1 (0.49) DYRK1AGSK3BWNT1CLK2CLK3
SCHEMBL18494630 0.65 WNT1 (0.48) DYRK1AWNT1CLK2CLK3
SCHEMBL18441698 0.64 WNT1 (0.61) DYRK1AGSK3BWNT1CLK2CLK3
SCHEMBL18443277 0.63 WNT1 (0.45) DYRK1AGSK3BWNT1CLK2CLK3
SCHEMBL7119935 0.63 RIPK2 (0.41) TTK
SCHEMBL18446957 0.62 WNT1 (0.57) DYRK1AWNT1CLK2CLK3
SCHEMBL28996272 0.62 BCHE (0.42) ALDH1A1TP53
SCHEMBL6754326 0.62 MAP4K4 (0.49) DYRK1ATTKCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001087845-A2 N-CONTAINING HETEROCYCLIC COMPOUNDS AND THEIR USE AS 5-HT ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-22 WO disclosed