SCHEMBL7984443

SCHEMBL7984443

CCCCCCCC#CC(SC(C#CCCCCCCC)c1ccccc1OC(C)=O)c1ccccc1OC(C)=O

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.58
PPARG P37231 2/20 0.43
PPARA Q07869 2/20 0.43
CYSLTR2 Q9NS75 2/20 0.42
CYSLTR1 Q9Y271 2/20 0.42
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7996233 1.00 PTGS2 (0.58) PTGS2PPARGPPARACYSLTR2CYSLTR1
SCHEMBL7996163 0.99 PTGS2 (0.59) PTGS2PPARGPPARACYSLTR2CYSLTR1
SCHEMBL3842936 0.95 PTGS2 (0.63) PTGS2PPARGPPARA
SCHEMBL6534900 0.90 PTGS2 (0.55) PTGS2
SCHEMBL7998377 0.85 PTGS2 (0.52) PTGS2PPARGPPARACYSLTR2CYSLTR1
SCHEMBL6535165 0.84 PTGS2 (0.53) PTGS2
SCHEMBL8001950 0.84 PTGS2 (0.60) PTGS2PPARGPPARACYSLTR2CYSLTR1
SCHEMBL7998114 0.84 PTGS2 (0.56) PTGS2PPARGPPARACYSLTR2CYSLTR1
SCHEMBL7996240 0.84 PTGS2 (0.56) PTGS2PPARGPPARACYSLTR2CYSLTR1
SCHEMBL7984449 0.84 PTGS2 (0.56) PTGS2PPARGPPARACYSLTR2CYSLTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6284918-B1 ENZYME INHIBITORS VANDERBILT UNIVERSITY 2001-09-04 US claimed
US-6284918-B1 ENZYME INHIBITORS VANDERBILT UNIVERSITY 2001-09-04 US disclosed