SCHEMBL7984449

SCHEMBL7984449

CCCCCCCC#CC(S)c1ccccc1OC(C)=O

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.56
PPARG P37231 2/20 0.43
PPARA Q07869 2/20 0.43
S1PR1 P21453 1/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CYSLTR2 Q9NS75 1/20 0.41
CYSLTR1 Q9Y271 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7998114 1.00 PTGS2 (0.56) PTGS2PPARGPPARAS1PR1CYP3A4
SCHEMBL7996240 1.00 PTGS2 (0.56) PTGS2PPARGPPARAS1PR1CYP3A4
SCHEMBL7996168 0.99 PTGS2 (0.57) PTGS2PPARGPPARAS1PR1CYP3A4
SCHEMBL3842942 0.95 PTGS2 (0.61) PTGS2PPARGPPARA
SCHEMBL6534904 0.90 PTGS2 (0.53) PTGS2
SCHEMBL7994632 0.86 PTGS2 (0.51) PTGS2PPARGPPARAS1PR1CYP3A4
SCHEMBL7998381 0.85 PTGS2 (0.50) PTGS2PPARGPPARAS1PR1CYP3A4
SCHEMBL6535172 0.84 PTGS2 (0.51) PTGS2CYP2C9
SCHEMBL7984443 0.84 PTGS2 (0.58) PTGS2PPARGPPARACYP3A4CYP2C9
SCHEMBL7996233 0.84 PTGS2 (0.58) PTGS2PPARGPPARACYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6284918-B1 ENZYME INHIBITORS VANDERBILT UNIVERSITY 2001-09-04 US claimed
US-6284918-B1 ENZYME INHIBITORS VANDERBILT UNIVERSITY 2001-09-04 US disclosed