SCHEMBL7984576

SCHEMBL7984576

O=C1Nc2ccc(C(=O)O)cc2/C1=C(/Nc1ccc(Cl)cc1)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.45
GSK3B P49841 5/20 0.42
PAK4 O96013 1/20 0.42
LRRK2 Q5S007 2/20 0.42
PDPK1 O15530 1/20 0.41
JAK3 P52333 1/20 0.41
TLK2 Q86UE8 1/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
CNR1 P21554 1/20 0.39
ALDH1A1 P00352 1/20 0.39
EPHX1 P07099 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7984532 0.89 RAB9A (0.49) KDRPAK4LRRK2PDPK1KMT2A
SCHEMBL7982075 0.89 PAK4 (0.43) KDRGSK3BPAK4LRRK2NPC1
SCHEMBL6980872 0.89 PAK4 (0.43) KDRGSK3BPAK4LRRK2NPC1
SCHEMBL7985455 0.88 JAK3 (0.44) KDRPAK4LRRK2PDPK1JAK3
SCHEMBL6982836 0.88 JAK3 (0.44) KDRPAK4LRRK2PDPK1JAK3
SCHEMBL8192969 0.87 HTT (0.45) KDRPAK4LRRK2JAK3KMT2A
SCHEMBL4493857 0.86 PLK1 (0.46) KDRKMT2AMEN1
SCHEMBL4493853 0.86 PLK1 (0.46) KDRKMT2AMEN1
SCHEMBL7088642 0.86 PDPK1 (0.44) KDRGSK3BLRRK2PDPK1KMT2A
SCHEMBL7972055 0.86 PDPK1 (0.44) KDRGSK3BLRRK2PDPK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6169106-B1 ANTITUMOUR AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-01-02 US disclosed