SCHEMBL7984532

SCHEMBL7984532

COC(=O)c1ccc2c(c1)/C(=C(/Nc1ccc(Cl)cc1)c1ccccc1)C(=O)N2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.49
NPC1 O15118 2/20 0.49
MAPT P10636 2/20 0.49
PDPK1 O15530 1/20 0.44
AURKA O14965 1/20 0.44
RAF1 P04049 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43
PSEN1 P49768 1/20 0.43
PSEN2 P49810 1/20 0.43
APH1B Q8WW43 1/20 0.43
NCSTN Q92542 1/20 0.43
APH1A Q96BI3 1/20 0.43
PSENEN Q9NZ42 1/20 0.43
KDR P35968 2/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
PLAU P00749 1/20 0.41
LRRK2 Q5S007 1/20 0.41
PTPN1 P18031 1/20 0.41
CNR1 P21554 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7987801 0.92 PDPK1 (0.48) RAB9ANPC1MAPTPDPK1AURKA
SCHEMBL2123765 0.92 RAB9A (0.49) RAB9ANPC1MAPTNPSR1PSEN1
SCHEMBL2123767 0.92 RAB9A (0.49) RAB9ANPC1MAPTNPSR1PSEN1
SCHEMBL7984576 0.89 KDR (0.45) RAB9ANPC1PDPK1NPSR1KDR
SCHEMBL6980872 0.88 PAK4 (0.43) RAB9ANPC1MAPTNPSR1KDR
SCHEMBL7982075 0.88 PAK4 (0.43) RAB9ANPC1MAPTNPSR1KDR
SCHEMBL7224171 0.87 MAPT (0.47) RAB9ANPC1MAPTPDPK1AURKA
SCHEMBL7985455 0.87 JAK3 (0.44) RAB9ANPC1PDPK1KDRKMT2A
SCHEMBL6982836 0.87 JAK3 (0.44) RAB9ANPC1PDPK1KDRKMT2A
SCHEMBL7085728 0.85 PTPN1 (0.44) RAB9ANPC1MAPTPDPK1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6169106-B1 ANTITUMOUR AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-01-02 US disclosed