SCHEMBL7984825

SCHEMBL7984825

CN(C)Cc1ccc(N/C(=C2\C(=O)Nc3ccc(C(=O)O)cc32)c2ccccc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.41
LTA4H P09960 3/20 0.38
SLC2A1 P11166 1/20 0.38
CYP3A4 P08684 2/20 0.38
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
LSS P48449 1/20 0.37
PDPK1 O15530 2/20 0.37
JAK3 P52333 1/20 0.37
TLK2 Q86UE8 1/20 0.37
SRC P12931 1/20 0.37
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
CYP2C19 P33261 1/20 0.36
PAK4 O96013 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4611892 0.93 ROCK2 (0.40) ROCK2SLC2A1PDPK1JAK3TLK2
SCHEMBL4611898 0.93 ROCK2 (0.40) ROCK2SLC2A1PDPK1JAK3TLK2
SCHEMBL14587215 0.93 ROCK2 (0.40) ROCK2SLC2A1PDPK1JAK3TLK2
SCHEMBL8186883 0.92 ROCK2 (0.48) ROCK2SLC2A1CYP3A4HDAC3HDAC1
SCHEMBL8186879 0.92 ROCK2 (0.48) ROCK2SLC2A1CYP3A4HDAC3HDAC1
SCHEMBL6984575 0.92 JAK3 (0.42) ROCK2SLC2A1CYP3A4HDAC3HDAC1
SCHEMBL6984569 0.92 JAK3 (0.42) ROCK2SLC2A1CYP3A4HDAC3HDAC1
SCHEMBL3157925 0.92 ROCK2 (0.43) ROCK2LTA4HSLC2A1CYP3A4HDAC3
SCHEMBL3157931 0.92 ROCK2 (0.43) ROCK2LTA4HSLC2A1CYP3A4HDAC3
SCHEMBL7981209 0.91 PDPK1 (0.41) ROCK2CYP3A4PDPK1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6169106-B1 ANTITUMOUR AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-01-02 US disclosed