SCHEMBL7985237

SCHEMBL7985237

COc1cccc(C(CN2CCCC2)N(C)C(=O)Cc2ccccc2[N+](=O)[O-])c1

nearest known ligand 0.78

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 17/20 0.78
CYP2D6 P10635 4/20 0.55
SIGMAR1 Q99720 1/20 0.53
OPRD1 P41143 5/20 0.53
OPRM1 P35372 4/20 0.53
CYP3A4 P08684 2/20 0.52
TSHR P16473 2/20 0.52
CYP2C19 P33261 1/20 0.52
CYP1A2 P05177 1/20 0.51
THPO P40225 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6479790 1.00 OPRK1 (0.78) OPRK1CYP2D6SIGMAR1OPRD1OPRM1
SCHEMBL6479796 1.00 OPRK1 (0.78) OPRK1CYP2D6SIGMAR1OPRD1OPRM1
SCHEMBL5630305 0.88 OPRK1 (0.82) OPRK1CYP2D6SIGMAR1OPRD1OPRM1
SCHEMBL5629262 0.88 OPRK1 (1.00) OPRK1CYP2D6SIGMAR1OPRD1OPRM1
SCHEMBL8459482 0.88 OPRK1 (1.00) OPRK1CYP2D6SIGMAR1OPRD1OPRM1
SCHEMBL6480069 0.85 OPRK1 (0.76) OPRK1CYP2D6OPRD1OPRM1CYP3A4
SCHEMBL7722061 0.85 OPRK1 (0.76) OPRK1CYP2D6OPRD1OPRM1CYP3A4
SCHEMBL6479482 0.85 OPRK1 (0.76) OPRK1CYP2D6OPRD1OPRM1CYP3A4
SCHEMBL10434997 0.83 OPRK1 (0.86) OPRK1CYP2D6SIGMAR1OPRD1OPRM1
SCHEMBL10434613 0.83 OPRK1 (0.82) OPRK1CYP2D6SIGMAR1OPRD1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6239154-B1 ARYLACETAMIDES, AGONISTS AT KAPPA OPIOID RECEPTORS. ADOLOR CORPORATION 2001-05-29 US disclosed
US-6057323-A PIPERAZINE DERIVATIVES ADOLOR CORPORATION (US) 2000-05-02 US disclosed