SCHEMBL7985252

SCHEMBL7985252

CN1C(=O)c2ccccc2[N]c2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 3/20 0.53
CES1 P23141 2/20 0.53
DRD2 P14416 2/20 0.47
HTR6 P50406 2/20 0.47
CASP3 P42574 1/20 0.46
LRRK2 Q5S007 1/20 0.44
MAPT P10636 4/20 0.43
RAB9A P51151 2/20 0.43
MAPK1 P28482 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TRPA1 O75762 1/20 0.42
NPC1 O15118 1/20 0.42
MTOR P42345 1/20 0.42
EPHX2 P34913 2/20 0.41
APP P05067 1/20 0.41
SNCA P37840 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6013602 0.81 TTR (0.47) TTRCES1DRD2HTR6CASP3
SCHEMBL16127516 0.78 TTR (0.75) TTRCES1DRD2HTR6CASP3
SCHEMBL2354261 0.76 TTR (0.41) TTRCES1DRD2HTR6CASP3
SCHEMBL12059596 0.74 TTR (0.69) TTRCES1DRD2HTR6CASP3
SCHEMBL29511191 0.70 CASP3 (0.81) TTRCES1CASP3MAPTL3MBTL1
SCHEMBL28263 0.70 CASP3 (0.81) TTRCES1CASP3MAPTL3MBTL1
SCHEMBL126628 0.70 CES1 (1.00) TTRCES1CASP3RAB9ATRPA1
SCHEMBL30077375 0.70 TTR (0.69) TTRCES1DRD2HTR6CASP3
SCHEMBL13039623 0.70 TTR (0.69) TTRCES1DRD2HTR6CASP3
SCHEMBL28252336 0.70 CES1 (1.00) TTRCES1CASP3RAB9ATRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235730-B1 ANTICHOLESTEROL AGENT, ANTILIPEMIC AGENT JAPAN TOBACCO, INC. (JP) 2001-05-22 US claimed
EP-0970954-A1 3-PIPERIDYL-4-OXOQUINAZOLINE DERIVATIVES AND MEDICINCAL COMPOSITIONS CONTAINING THE SAME JAPAN TOBACCO INC. (JP) 2000-01-12 EP claimed
US-6235730-B1 ANTICHOLESTEROL AGENT, ANTILIPEMIC AGENT JAPAN TOBACCO, INC. (JP) 2001-05-22 US disclosed
EP-0970954-A1 3-PIPERIDYL-4-OXOQUINAZOLINE DERIVATIVES AND MEDICINCAL COMPOSITIONS CONTAINING THE SAME JAPAN TOBACCO INC. (JP) 2000-01-12 EP disclosed