SCHEMBL7985474

SCHEMBL7985474

c1ccc2c(c1)CN(C1CCNCC1)C2

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.50
HTR2A P28223 3/20 0.50
HTR2B P41595 2/20 0.46
HPGD P15428 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KCNH2 Q12809 2/20 0.42
HRH3 Q9Y5N1 2/20 0.42
CRBN Q96SW2 1/20 0.42
SLC18A3 Q16572 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
NAMPT P43490 1/20 0.42
PARP1 P09874 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12537066 0.90 HTR2C (0.46) HTR2CHTR2AHTR2BHPGDKMT2A
SCHEMBL14069048 0.88 HTR2C (0.46) HTR2CHTR2AHTR2BCRBNSLC18A3
SCHEMBL29501341 0.87 SLC18A3 (0.53) HTR2CHTR2AHTR2BHRH3SLC18A3
SCHEMBL2657988 0.87 SLC18A3 (0.53) HTR2CHTR2AHTR2BHRH3SLC18A3
Bromide SCHEMBL6423364 0.86 SLC18A3 (0.51) HTR2CHTR2AHTR2BHRH3SLC18A3
Hydrochloric Acid SCHEMBL5271851 0.86 SLC18A3 (0.51) HTR2CHTR2AHTR2BHPGDKMT2A
Hydrochloric Acid SCHEMBL29877056 0.86 SLC18A3 (0.51) HTR2CHTR2AHTR2BHPGDKMT2A
Hydrochloric Acid SCHEMBL16835555 0.86 SLC18A3 (0.51) HTR2CHTR2AHTR2BHPGDKMT2A
SCHEMBL11265606 0.84 HRH3 (0.53) KCNH2HRH3CRBNSLC18A3
SCHEMBL11639039 0.82 HTR2C (0.58) HTR2CHTR2AHTR2BHPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018144900-A1 SMALL MOLECULE ANTAGONISTS OF SUMO RELATED MODIFICATION OF CRMP2 AND USES THEREOF ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2018-08-09 WO disclosed
US-6235730-B1 ANTICHOLESTEROL AGENT, ANTILIPEMIC AGENT JAPAN TOBACCO, INC. (JP) 2001-05-22 US disclosed