SCHEMBL7986865

SCHEMBL7986865

COc1cccc(-c2cncc(-c3cn(CCCN4CCCCC4)c4cccnc34)c2)c1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.50
FLT1 P17948 2/20 0.50
FLT4 P35916 2/20 0.50
HRH3 Q9Y5N1 8/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
KMT2A Q03164 1/20 0.43
BACE1 P56817 1/20 0.41
GSK3B P49841 2/20 0.40
QPCT Q16769 2/20 0.40
KCNH2 Q12809 1/20 0.39
LTA4H P09960 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7551471 0.95 KDR (0.49) KDRFLT1FLT4HRH3KDM4E
SCHEMBL7550710 0.93 KDR (0.52) KDRFLT1FLT4GSK3BQPCT
SCHEMBL7986889 0.91 KDR (0.51) KDRFLT1FLT4HRH3GSK3B
SCHEMBL7556924 0.87 KDR (0.59) KDRFLT1FLT4HRH3GSK3B
SCHEMBL7554860 0.87 CYP1A2 (0.49) KDRFLT1FLT4ALDH1A1GSK3B
SCHEMBL7549925 0.86 KDR (0.67) KDRFLT1FLT4HRH3GSK3B
SCHEMBL7551303 0.86 KDR (0.52) KDRFLT1FLT4HRH3GSK3B
SCHEMBL7986847 0.85 KDR (0.50) KDRFLT1FLT4KDM4EALDH1A1
SCHEMBL7558444 0.85 KDR (0.57) KDRFLT1FLT4HRH3KDM4E
SCHEMBL7547677 0.85 KDR (0.49) KDRBACE1GSK3BQPCT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed