SCHEMBL7986847

SCHEMBL7986847

COc1ccc(-c2cncc(-c3cn(CCN4CCCCC4)c4cccnc34)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.50
FLT1 P17948 4/20 0.44
FLT4 P35916 4/20 0.44
CHRNB1 P11230 1/20 0.41
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNB3 Q05901 1/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
RCE1 Q9Y256 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
FLT3 P36888 1/20 0.39
MAPK14 Q16539 2/20 0.39
HSD17B10 Q99714 1/20 0.39
PDE10A Q9Y233 1/20 0.39
MCHR1 Q99705 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7986889 0.94 KDR (0.51) KDRFLT1FLT4CHRNB1CHRNB2
SCHEMBL7990494 0.92 KDR (0.51) KDRFLT1FLT4KDM4EALDH1A1
SCHEMBL7551471 0.91 KDR (0.49) KDRFLT1FLT4CHRNB1CHRNB2
SCHEMBL7548593 0.88 KDR (0.57) KDRFLT1FLT4SIGMAR1MAPK14
SCHEMBL7555532 0.87 KDR (0.52) KDRFLT1FLT4CHRNB1CHRNB2
SCHEMBL7551398 0.87 KDR (0.54) KDRFLT1FLT4CHRNB1CHRNB2
SCHEMBL7551721 0.87 CHRNB1 (0.39) KDRFLT1FLT4CHRNB1CHRNB2
SCHEMBL7986865 0.85 KDR (0.50) KDRFLT1FLT4KDM4EALDH1A1
SCHEMBL7555221 0.85 KDR (0.68) KDRFLT1FLT4FLT3MKNK2
SCHEMBL7554860 0.83 CYP1A2 (0.49) KDRFLT1FLT4ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed