SCHEMBL7986889

SCHEMBL7986889

COc1ccc(-c2cncc(-c3cn(CCCN4CCCCC4)c4cccnc34)c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.51
FLT1 P17948 3/20 0.51
FLT4 P35916 3/20 0.51
GSK3B P49841 6/20 0.43
QPCT Q16769 6/20 0.43
HTR3A P46098 5/20 0.41
HRH3 Q9Y5N1 2/20 0.40
KCNH2 Q12809 1/20 0.40
ACHE P22303 1/20 0.40
CHRNB1 P11230 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNB3 Q05901 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7986847 0.94 KDR (0.50) KDRFLT1FLT4HTR3ACHRNB1
SCHEMBL7551398 0.93 KDR (0.54) KDRFLT1FLT4GSK3BQPCT
SCHEMBL7986865 0.91 KDR (0.50) KDRFLT1FLT4GSK3BQPCT
SCHEMBL7556924 0.89 KDR (0.59) KDRFLT1FLT4GSK3BHRH3
SCHEMBL7987168 0.88 KDR (0.54) KDRFLT1FLT4GSK3BQPCT
SCHEMBL7990494 0.86 KDR (0.51) KDRFLT1FLT4GSK3B
SCHEMBL7554266 0.86 KDR (0.69) KDRFLT1FLT4GSK3BQPCT
SCHEMBL7551471 0.85 KDR (0.49) KDRFLT1FLT4HRH3CHRNB1
SCHEMBL7549825 0.84 KDR (0.51) KDRGSK3BQPCT
SCHEMBL7550710 0.84 KDR (0.52) KDRFLT1FLT4GSK3BQPCT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed