SCHEMBL7987650

SCHEMBL7987650

CCOC(=O)CC[C@@H](C(=O)OCC)n1sc2cc(NCc3ccc4ccc5nc(C)[nH]c(=O)c5c4c3)ccc2c1=O

nearest known ligand 0.78

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TYMS P04818 9/20 0.78
DHFR P00374 1/20 0.38
P2RX3 P56373 1/20 0.36
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
P2RY12 Q9H244 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6649605 0.88 TYMS (1.00) TYMSDHFR
SCHEMBL7990232 0.81 TYMS (0.78) TYMSDHFR
SCHEMBL7501783 0.81 TYMS (0.78) TYMSDHFR
SCHEMBL6654917 0.78 TYMS (0.60) TYMSDHFR
SCHEMBL6654911 0.78 TYMS (0.60) TYMSDHFR
SCHEMBL6446395 0.78 TYMS (0.77) TYMS
SCHEMBL6446404 0.78 TYMS (0.77) TYMS
SCHEMBL6447640 0.77 TYMS (0.52) TYMSDHFRPDE3BPDE3AP2RY12
SCHEMBL7258233 0.76 TYMS (0.73) TYMS
SCHEMBL9422199 0.74 TYMS (0.55) TYMSDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306865-B1 SYNTHASE INHIBITORS AND ANTITUMOR AGENTS GLAXO WELLCOME INC. 2001-10-23 US disclosed