SCHEMBL7990232

SCHEMBL7990232

CCOC(=O)CCC(C(=O)OCC)N1Cc2cc(NCc3ccc4ccc5nc(C)[nH]c(=O)c5c4c3)ccc2C1=O

nearest known ligand 0.78

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TYMS P04818 9/20 0.78
DHFR P00374 4/20 0.42
SLC19A1 P41440 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7501783 1.00 TYMS (0.78) TYMSDHFRSLC19A1
SCHEMBL6450938 0.91 TYMS (0.65) TYMSDHFRSLC19A1
SCHEMBL7258331 0.90 TYMS (0.69) TYMSDHFR
Osi-7904 SCHEMBL2195534 0.88 TYMS (1.00) TYMSDHFRSLC19A1
Osi-7904 SCHEMBL7207397 0.88 TYMS (1.00) TYMSDHFRSLC19A1
Osi-7904 SCHEMBL29389995 0.88 TYMS (1.00) TYMSDHFRSLC19A1
Osi-7904 SCHEMBL29692303 0.88 TYMS (1.00) TYMSDHFRSLC19A1
Osi-7904 SCHEMBL29692323 0.88 TYMS (1.00) TYMSDHFRSLC19A1
SCHEMBL7987650 0.81 TYMS (0.78) TYMSDHFR
SCHEMBL2638076 0.80 TYMS (0.81) TYMSDHFRSLC19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306865-B1 SYNTHASE INHIBITORS AND ANTITUMOR AGENTS GLAXO WELLCOME INC. 2001-10-23 US disclosed