SCHEMBL7987965

SCHEMBL7987965

COC(=O)c1cccc2c1c(-c1cncc(-c3cccc(OC)c3)c1)cn2CCN1CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.45
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
AVPR1B P47901 4/20 0.41
KCNH2 Q12809 1/20 0.41
HRH3 Q9Y5N1 5/20 0.41
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
FLT1 P17948 1/20 0.41
FLT4 P35916 1/20 0.41
MCL1 Q07820 1/20 0.40
BAD Q92934 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7549814 0.95 FLT1 (0.47) KDRKMT2AKDM4EALDH1A1AVPR1B
SCHEMBL7990656 0.93 CYP1A2 (0.48) KDRALDH1A1AVPR1BNPSR1FLT1
SCHEMBL7994209 0.92 KDR (0.46) KDRKMT2AKDM4EALDH1A1ROCK2
SCHEMBL7554912 0.91 KDR (0.50) KDRKMT2AHRH3FLT1FLT4
SCHEMBL7993627 0.90 KDR (0.45) KDRKMT2AAVPR1BHRH3FLT1
SCHEMBL7550186 0.89 KDR (0.49) KDRKMT2AKDM4EALDH1A1KCNH2
SCHEMBL7551275 0.88 KDR (0.47) KDRKMT2AKDM4EALDH1A1KCNH2
SCHEMBL7987156 0.87 KDR (0.46) KDRKMT2AKDM4EFLT1FLT4
SCHEMBL7549576 0.86 KDR (0.51) KDRKMT2AKDM4EALDH1A1HRH3
SCHEMBL7551621 0.86 KDR (0.64) KDRKMT2AFLT1FLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed