SCHEMBL7990656

SCHEMBL7990656

COC(=O)c1cccc2c1c(-c1cncc(-c3cccc(OC)c3)c1)cn2CCN1CCOCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
ALOX15 P16050 1/20 0.48
HIF1A Q16665 1/20 0.48
HSD17B10 Q99714 1/20 0.48
FLT1 P17948 1/20 0.46
FLT4 P35916 1/20 0.46
KDR P35968 1/20 0.46
CNR1 P21554 3/20 0.46
CNR2 P34972 3/20 0.45
ALDH1A1 P00352 3/20 0.44
USP2 O75604 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
GSK3B P49841 1/20 0.43
DYRK1A Q13627 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7987965 0.93 KDR (0.45) FLT1FLT4KDRALDH1A1AVPR1B
SCHEMBL7976639 0.93 FLT1 (0.47) HSD17B10FLT1FLT4KDRCNR1
SCHEMBL7508991 0.92 CNR1 (0.51) FLT1FLT4KDRCNR1CNR2
SCHEMBL7986724 0.90 FLT1 (0.46) TP53FLT1FLT4KDRCNR1
SCHEMBL7550186 0.88 KDR (0.49) FLT1FLT4KDRALDH1A1GSK3B
SCHEMBL7549814 0.88 FLT1 (0.47) FLT1FLT4KDRALDH1A1AVPR1B
SCHEMBL7991040 0.88 FLT1 (0.47) TP53FLT1FLT4KDRCNR1
SCHEMBL7513681 0.86 KDR (0.65) FLT1FLT4KDRCNR1CNR2
SCHEMBL7553606 0.85 KDR (0.49) CYP1A2CYP3A4CYP2D6LMNATP53
SCHEMBL7994209 0.85 KDR (0.46) CYP1A2CYP2D6ALOX15FLT1FLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed