SCHEMBL7988229

SCHEMBL7988229

CCOC(=O)Cn1cc2c(n1)CCN(C(=O)[C@H](Cc1ccc(OCc3ccccc3)cc1)NC(=O)OC(C)(C)C)C2

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.51
HRH2 P25021 1/20 0.46
HRH1 P35367 1/20 0.46
P2RX7 Q99572 8/20 0.45
YAP1 P46937 2/20 0.44
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
BCL2 P10415 1/20 0.44
PTPN1 P18031 3/20 0.44
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7974848 0.93 ADORA1 (0.56) ADORA1HRH2HRH1P2RX7ITGB3
SCHEMBL7988287 0.88 ADORA1 (0.48) ADORA1P2RX7ITGB3ITGA2BKMT2A
SCHEMBL7989135 0.88 ADORA1 (0.48) ADORA1HRH2HRH1P2RX7ITGB3
SCHEMBL7988765 0.87 ADORA1 (0.46) ADORA1HRH2HRH1P2RX7ITGB3
SCHEMBL7986800 0.85 ITGB3 (0.44) ADORA1HRH2HRH1P2RX7YAP1
SCHEMBL7988313 0.85 ITGB3 (0.59) ADORA1HRH2HRH1P2RX7ITGB3
SCHEMBL7986455 0.82 ADORA1 (0.43) ADORA1HRH2HRH1ITGB3ITGA2B
SCHEMBL7986565 0.81 ADORA1 (0.55) ADORA1HRH2HRH1P2RX7YAP1
SCHEMBL7988835 0.81 KMT2A (0.42) ADORA1HRH2HRH1ITGB3ITGA2B
SCHEMBL2583794 0.80 P2RX7 (0.63) ADORA1HRH2HRH1P2RX7YAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265418-B1 ANTICOAGULANTS UBE INDUSTRIES, LTD. (JP) 2001-07-24 US disclosed
EP-1020467-A1 N-ACYLAMINO ACID AMIDE COMPOUNDS AND INTERMEDIATES FOR PREPARATION THEREOF UBE INDUSTRIES LIMITED (JP) 2000-07-19 EP disclosed