SCHEMBL7989374

SCHEMBL7989374

c1csc(CCCSc2nsnc2[C@H]2CN3CCC[C@H]2C3)c1

nearest known ligand 0.74

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 2/20 0.56
CHRM2 P08172 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7810793 1.00 CHRM1 (0.56) CHRM1CHRM2
Oxalic Acid SCHEMBL7810636 0.95 CHRM1 (0.54) CHRM1CHRM2
Oxalic Acid SCHEMBL7953188 0.95 CHRM1 (0.54) CHRM1CHRM2
SCHEMBL7818869 0.94 CHRM2 (0.54) CHRM1CHRM2
Oxalic Acid SCHEMBL7821928 0.91 CHRM2 (0.52) CHRM1CHRM2
SCHEMBL7818023 0.89 CHRM2 (0.48) CHRM2
SCHEMBL7810907 0.85 CHRM2 (0.65) CHRM1CHRM2
SCHEMBL8196540 0.84 CHRM1 (0.60) CHRM1CHRM2
SCHEMBL8197694 0.83 CHRM1 (0.59) CHRM1CHRM2
Oxalic Acid SCHEMBL7811971 0.82 CHRM2 (0.61) CHRM1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6271229-B1 ADMINISTERING A 1,2,5-OXADIAZOLE COMPOUND OR 1,2,5-THIADIAZOLE COMPOUND NOVO NORDISK A/S (DK) 2001-08-07 US claimed
EP-0873124-A1 A METHOD OF TREATING HYPERCHOLESTEROLEMIA AND RELATED DISORDERS NOVO NORDISK A/S (DK) 1998-10-28 EP claimed
US-5750538-A 1,2,5-THIADIAZOL-4-YL-1-AZABICYCLIC DERIVATIVES NOVO NORDISK A/S (DK) 1998-05-12 US claimed
US-5710151-A ADMINISTERING A THIADIAZOLE OR AN OXADIAZOLE DERIVATIVE TO A SUBJECT MUHLHAUSER MARK A (US) 1998-01-20 US claimed
WO-1997025043-A1 A METHOD OF TREATING HYPERCHOLESTEROLEMIA AND RELATED DISORDERS NOVO NORDISK A/S (DK) 1997-07-17 WO claimed
WO-1996014316-A1 A METHOD OF TREATING URINARY BLADDER DYSFUNCTIONS NOVO NORDISK A/S (DK) 1996-05-17 WO claimed
EP-0709093-B1 Method for treating anxiety using an azabicyclic oxadiazole or thiadiazole compound LILLY CO ELI (US) 2000-04-05 EP disclosed
US-5750538-A 1,2,5-THIADIAZOL-4-YL-1-AZABICYCLIC DERIVATIVES NOVO NORDISK A/S (DK) 1998-05-12 US disclosed
US-5726193-A OXADIAZOLE- AND THIADIAZOLE-SUBSTITUTED AZABICYCLOALKANES ELI LILLY AND COMPANY (US) 1998-03-10 US disclosed
EP-0709093-A2 Method for treating anxiety using an azabicyclic oxadiazole or thiadiazole compound ELI LILLY AND COMPANY (US) 1996-05-01 EP disclosed
US-5484794-A THIA- OR OXA-DIAZOLE COMPOUNDS ELI LILLY AND COMPANY (US) 1996-01-16 US disclosed