SCHEMBL7810907

SCHEMBL7810907

c1ccc(CCCSc2nsnc2C2CN3CCCC2C3)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.65
CHRM1 P11229 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL7811971 0.96 CHRM2 (0.61) CHRM2CHRM1
SCHEMBL7810578 0.93 CHRM2 (0.64) CHRM2CHRM1
Oxalic Acid SCHEMBL7819179 0.91 CHRM2 (0.58) CHRM2CHRM1
SCHEMBL7818477 0.89 CHRM2 (0.58) CHRM2CHRM1
SCHEMBL8196540 0.87 CHRM1 (0.60) CHRM2CHRM1
SCHEMBL7989374 0.85 CHRM1 (0.56) CHRM2CHRM1
SCHEMBL7810793 0.85 CHRM1 (0.56) CHRM2CHRM1
SCHEMBL9544481 0.85 CHRM1 (0.58) CHRM2CHRM1
Oxalic Acid SCHEMBL7953188 0.83 CHRM1 (0.54) CHRM2CHRM1
Oxalic Acid SCHEMBL7810636 0.83 CHRM1 (0.54) CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6271229-B1 ADMINISTERING A 1,2,5-OXADIAZOLE COMPOUND OR 1,2,5-THIADIAZOLE COMPOUND NOVO NORDISK A/S (DK) 2001-08-07 US claimed
EP-0714394-B1 ANTIPSYCHOTIC METHOD WITH THIADIAZOLE AND OXADIAZOLE DERIVATIVES NOVO NORDISK AS (DK) 2001-06-20 EP claimed
EP-0544779-B1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK AS (DK) 1998-12-02 EP claimed
EP-0873124-A1 A METHOD OF TREATING HYPERCHOLESTEROLEMIA AND RELATED DISORDERS NOVO NORDISK A/S (DK) 1998-10-28 EP claimed
EP-0866702-A1 METHOD FOR TREATING PAIN ELI LILLY AND COMPANY (US) 1998-09-30 EP claimed
WO-1997020556-A9 METHOD FOR TREATING PAIN 1997-10-02 WO claimed
EP-0790995-A1 A METHOD OF TREATING URINARY BLADDER DYSFUNCTIONS NOVO NORDISK A/S (DK) 1997-08-27 EP claimed
WO-1997025043-A1 A METHOD OF TREATING HYPERCHOLESTEROLEMIA AND RELATED DISORDERS NOVO NORDISK A/S (DK) 1997-07-17 WO claimed
WO-1997020556-A1 METHOD FOR TREATING PAIN ELI LILLY AND COMPANY (US) 1997-06-12 WO claimed
US-5574043-A ALZHEIMERS, GLAUCOMA, ANALGESIC NOVO NORDISK A/S (DK) 1996-11-12 US claimed
EP-0735869-A1 A METHOD OF TREATING GASTROINTESTINAL MOTILITY DISORDERS NOVO NORDISK A/S (DK) 1996-10-09 EP claimed
WO-1996014316-A1 A METHOD OF TREATING URINARY BLADDER DYSFUNCTIONS NOVO NORDISK A/S (DK) 1996-05-17 WO claimed
EP-0687266-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1995-12-20 EP claimed
WO-1995017180-A1 A METHOD OF TREATING GASTROINTESTINAL MOTILITY DISORDERS NOVO NORDISK A/S (DK) 1995-06-29 WO claimed
WO-1994020496-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1994-09-15 WO claimed
EP-0544779-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1993-06-09 EP claimed
WO-1992003433-A1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1992-03-05 WO claimed
CN-1292796-A METH1 and METH2 polynucleotides and polypeptides BETH ISRAEL DICKNY MEDICAL CT (US) 2001-04-25 CN disclosed
EP-0709093-A2 Method for treating anxiety using an azabicyclic oxadiazole or thiadiazole compound ELI LILLY AND COMPANY (US) 1996-05-01 EP disclosed
US-5484794-A THIA- OR OXA-DIAZOLE COMPOUNDS ELI LILLY AND COMPANY (US) 1996-01-16 US disclosed