SCHEMBL79894

SCHEMBL79894

O=C(N[C@H](CO)CC(=O)N(Cc1cccc(Cl)c1Cl)C1CC1)OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.47
SLC6A2 P23975 4/20 0.47
REN P00797 3/20 0.43
CYP3A4 P08684 3/20 0.42
SLC6A3 Q01959 2/20 0.42
CYP2D6 P10635 1/20 0.42
KCNH2 Q12809 1/20 0.42
CASP1 P29466 3/20 0.42
CTRB1 P17538 2/20 0.40
GHSR Q92847 1/20 0.40
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
PTPN7 P35236 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRK1 P41145 1/20 0.39
HTT P42858 1/20 0.39
DUSP3 P51452 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78618 0.76 SLC6A4 (0.51) SLC6A4SLC6A2RENCYP3A4SLC6A3
SCHEMBL65338 0.75 SLC6A4 (0.58) SLC6A4SLC6A2RENCYP3A4SLC6A3
SCHEMBL79378 0.75 SLC6A4 (0.64) SLC6A4SLC6A2RENCYP3A4SLC6A3
SCHEMBL5483040 0.72 MEN1 (0.52) SLC6A4SLC6A2CYP3A4GHSRMEN1
SCHEMBL10058367 0.72 CTRB1 (0.54) CYP3A4CTRB1MEN1LMNAKMT2A
SCHEMBL264008 0.70 CTRB1 (0.61) CASP1CTRB1
SCHEMBL553905 0.70 CTRB1 (0.61) CASP1CTRB1
SCHEMBL553906 0.70 CTRB1 (0.61) CASP1CTRB1
SCHEMBL4829896 0.70 CTRB1 (0.68) CTRB1ALDH1A1LMNASMN1; SMN2
SCHEMBL24324242 0.69 CTRB1 (0.53) CYP3A4CYP2D6CASP1CTRB1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed