SCHEMBL7989440

SCHEMBL7989440

CC(C)COc1cccc(CCN)c1

nearest known ligand 0.62

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 8/20 0.62
ACHE P22303 3/20 0.50
MAOB P27338 2/20 0.49
DRD2 P14416 1/20 0.44
DRD1 P21728 1/20 0.44
AOC3 Q16853 1/20 0.44
SIRT2 Q8IXJ6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31538932 0.86 MAOB (0.49) TAAR1MAOBSIRT2
SCHEMBL20825574 0.86 MAOB (0.49) TAAR1MAOBSIRT2
SCHEMBL327462 0.85 PPARA (0.46) TAAR1AOC3
SCHEMBL28032739 0.84 TAAR1 (0.58) TAAR1ACHEMAOB
SCHEMBL18183459 0.83 TAAR1 (0.57) TAAR1ACHEMAOBDRD2DRD1
SCHEMBL11806920 0.83 FAAH (0.42) TAAR1DRD2AOC3SIRT2
SCHEMBL8048495 0.83 CYP4F2 (0.61) TAAR1AOC3SIRT2
SCHEMBL8048492 0.83 NR1H4 (0.46) TAAR1AOC3SIRT2
SCHEMBL146849 0.81 TAAR1 (0.68) TAAR1ACHEMAOBDRD2DRD1
SCHEMBL30820845 0.81 TAAR1 (0.68) TAAR1ACHEMAOBDRD2DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001055117-A1 NOVEL ISOQUINOLINE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES SERVIER (FR) 2001-08-02 WO disclosed
US-5231181-A PROCESS FOR THE PREPARATION OF (8AS,12AS,13AS)-DECAHYDROISOQUINO ((2,1-G) (1,6)-NAPHTHYRIDIN-8-ONE DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1993-07-27 US disclosed
EP-0505183-A2 Process for the preparation of (8aS,12aS,13aS)-decahydroisoquino[2,1-g][1,6]-naphthyridin-8-one derivatives SYNTEX (U.S.A.) INC. (US) 1992-09-23 EP disclosed