SCHEMBL7990694

SCHEMBL7990694

COc1cccc2c(-c3cncc(-c4ccccc4)c3)cn(CC(C)CN(C)C)c12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.56
FLT1 P17948 1/20 0.56
FLT4 P35916 1/20 0.56
CNR2 P34972 2/20 0.41
HTR6 P50406 1/20 0.37
BRD9 Q9H8M2 3/20 0.35
BRD7 Q9NPI1 3/20 0.35
BRD4 O60885 1/20 0.35
BRD2 P25440 1/20 0.35
PRKACA P17612 1/20 0.35
PRKACG P22612 1/20 0.35
PRKACB P22694 1/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
KCNH2 Q12809 3/20 0.34
HCRTR1 O43613 2/20 0.34
HCRTR2 O43614 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7545417 0.93 KDR (0.52) KDRFLT1FLT4CNR2HTR6
SCHEMBL7504851 0.92 KDR (0.51) KDRFLT1FLT4CNR2HTR6
SCHEMBL7547229 0.92 KDR (0.51) KDRFLT1FLT4CNR2HTR6
SCHEMBL7546769 0.91 KDR (0.51) KDRFLT1FLT4CNR2HTR6
SCHEMBL7990474 0.88 KDR (0.71) KDRFLT1FLT4CNR2
SCHEMBL7549333 0.86 KDR (0.43) KDRFLT1FLT4CNR2HTR6
SCHEMBL7550357 0.83 KDR (0.78) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7549622 0.82 KDR (0.55) KDRFLT1FLT4CNR2HTR6
SCHEMBL7977281 0.81 KDR (0.61) KDRFLT1FLT4HTR6PRKACA
SCHEMBL7547790 0.80 KDR (0.68) KDRFLT1FLT4BRD4PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed