SCHEMBL7990934

SCHEMBL7990934

COc1cccc(-c2cncc(-c3cn(CCN4CCOCC4)c4ccccc34)c2)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.66
FLT1 P17948 3/20 0.66
FLT4 P35916 3/20 0.66
MKNK2 Q9HBH9 1/20 0.51
GSK3B P49841 3/20 0.50
CYP1A2 P05177 3/20 0.49
CYP3A4 P08684 3/20 0.49
CYP2D6 P10635 3/20 0.49
HSD17B10 Q99714 2/20 0.49
LMNA P02545 1/20 0.49
TP53 P04637 1/20 0.49
ALOX15 P16050 1/20 0.49
HIF1A Q16665 1/20 0.49
USP2 O75604 2/20 0.48
CLK4 Q9HAZ1 2/20 0.48
CYP2C19 P33261 1/20 0.48
ALDH1A1 P00352 3/20 0.47
NFATC1 O95644 1/20 0.46
DYRK1A Q13627 1/20 0.46
QPCT Q16769 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7990446 0.93 KDR (0.56) KDRFLT1FLT4MKNK2GSK3B
SCHEMBL7554226 0.91 KDR (0.66) KDRFLT1FLT4MKNK2GSK3B
SCHEMBL7990662 0.90 KDR (0.68) KDRFLT1FLT4MKNK2GSK3B
SCHEMBL7976794 0.89 KDR (0.53) KDRFLT1FLT4MKNK2GSK3B
SCHEMBL7986681 0.89 KDR (0.53) KDRFLT1FLT4MKNK2GSK3B
SCHEMBL7991015 0.88 KDR (0.59) KDRFLT1FLT4MKNK2GSK3B
SCHEMBL7976879 0.87 KDR (0.50) KDRFLT1FLT4MKNK2GSK3B
SCHEMBL7502516 0.87 KDR (0.77) KDRFLT1FLT4GSK3BNFATC1
SCHEMBL7986885 0.87 KDR (0.51) KDRFLT1FLT4MKNK2GSK3B
SCHEMBL7554860 0.86 CYP1A2 (0.49) KDRFLT1FLT4MKNK2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed