SCHEMBL7976879

SCHEMBL7976879

COc1cccc(-c2cncc(-c3cn(CCN4CCOCC4)c4c(OC)cccc34)c2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.50
FLT1 P17948 1/20 0.50
FLT4 P35916 1/20 0.50
CYP1A2 P05177 3/20 0.48
CYP3A4 P08684 3/20 0.48
CYP2D6 P10635 3/20 0.48
HSD17B10 Q99714 2/20 0.48
LMNA P02545 1/20 0.48
TP53 P04637 1/20 0.48
ALOX15 P16050 1/20 0.48
HIF1A Q16665 1/20 0.48
ALDH1A1 P00352 3/20 0.45
USP2 O75604 2/20 0.45
CLK4 Q9HAZ1 2/20 0.45
CYP2C19 P33261 1/20 0.45
CNR2 P34972 5/20 0.44
TSHR P16473 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CHEK1 O14757 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7988115 0.92 KDR (0.49) KDRFLT1FLT4CYP1A2CYP3A4
SCHEMBL7987655 0.92 KDR (0.51) KDRFLT1FLT4CYP1A2CYP3A4
SCHEMBL7990350 0.92 KDR (0.55) KDRFLT1FLT4CYP1A2CYP3A4
SCHEMBL7990490 0.90 KDR (0.49) KDRFLT1FLT4CYP2D6LMNA
SCHEMBL7990572 0.87 KDR (0.50) KDRFLT1FLT4CYP1A2CYP3A4
SCHEMBL7990934 0.87 KDR (0.66) KDRFLT1FLT4CYP1A2CYP3A4
SCHEMBL7555367 0.86 KDR (0.51) KDRFLT1FLT4ALDH1A1CNR2
SCHEMBL7556041 0.86 KDR (0.53) KDRFLT1FLT4CYP1A2CYP3A4
SCHEMBL7550119 0.86 CNR2 (0.40) KDRFLT1FLT4CYP1A2CYP3A4
SCHEMBL7987725 0.86 KDR (0.70) KDRFLT1FLT4CYP2D6CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed