SCHEMBL7992050

SCHEMBL7992050

CCOC(=O)Cc1cc2c(s1)CCN(C(=O)[C@H](Cc1ccncc1)NC(=O)OC(C)(C)C)C2

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.52
HRH2 P25021 2/20 0.44
HRH1 P35367 2/20 0.44
KMT2A Q03164 3/20 0.40
HCRTR2 O43614 4/20 0.38
MAPK1 P28482 1/20 0.38
PTPRB P23467 1/20 0.38
ROCK2 O75116 2/20 0.36
ACE P12821 1/20 0.35
PARP1 P09874 1/20 0.35
HCRTR1 O43613 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7986065 0.91 ADORA1 (0.51) ADORA1HRH2HRH1KMT2AHCRTR2
SCHEMBL7986071 0.91 ADORA1 (0.52) ADORA1KMT2AHCRTR2MAPK1PTPRB
SCHEMBL7992666 0.91 ADORA1 (0.56) ADORA1HRH2HRH1KMT2AHCRTR2
SCHEMBL7975232 0.89 ADORA1 (0.51) ADORA1HRH2HRH1KMT2A
SCHEMBL7985559 0.88 ADORA1 (0.50) ADORA1KMT2AHCRTR2MAPK1PTPRB
SCHEMBL7985657 0.88 ADORA1 (0.50) ADORA1KMT2AHCRTR2MAPK1PTPRB
SCHEMBL7986565 0.86 ADORA1 (0.55) ADORA1HRH2HRH1KMT2A
SCHEMBL7975386 0.86 ADORA1 (0.53) ADORA1HRH2HRH1KMT2AHCRTR2
SCHEMBL7989016 0.85 ADORA1 (0.54) ADORA1KMT2AHCRTR2MAPK1
SCHEMBL7986391 0.85 ADORA1 (0.47) ADORA1HRH2HRH1KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265418-B1 ANTICOAGULANTS UBE INDUSTRIES, LTD. (JP) 2001-07-24 US disclosed
EP-1020467-A1 N-ACYLAMINO ACID AMIDE COMPOUNDS AND INTERMEDIATES FOR PREPARATION THEREOF UBE INDUSTRIES LIMITED (JP) 2000-07-19 EP disclosed