SCHEMBL7994167

SCHEMBL7994167

COC(=O)CN1CN(c2ccccc2)C2(CCN(Cc3ccc(N(C)C)cc3)CC2)C1=O

nearest known ligand 0.74

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.74
CYP3A4 P08684 1/20 0.74
CYP2D6 P10635 1/20 0.74
CYP2C9 P11712 1/20 0.74
KMT2A Q03164 1/20 0.74
OPRL1 P41146 12/20 0.66
OPRM1 P35372 10/20 0.60
OPRK1 P41145 10/20 0.60
BDKRB2 P30411 1/20 0.52
OPRD1 P41143 9/20 0.51
DRD2 P14416 1/20 0.51
DRD3 P35462 1/20 0.51
NPC1L1 Q9UHC9 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7995842 0.89 CYP2D6 (0.80) MEN1CYP3A4CYP2D6CYP2C9KMT2A
SCHEMBL7759170 0.89 MEN1 (0.77) MEN1CYP3A4CYP2D6CYP2C9KMT2A
SCHEMBL7995949 0.86 MEN1 (0.79) MEN1CYP3A4CYP2D6CYP2C9KMT2A
SCHEMBL7760219 0.85 MEN1 (0.72) MEN1CYP3A4CYP2D6CYP2C9KMT2A
SCHEMBL7992840 0.85 MEN1 (1.00) MEN1CYP3A4CYP2D6CYP2C9KMT2A
SCHEMBL29789407 0.85 MEN1 (1.00) MEN1CYP3A4CYP2D6CYP2C9KMT2A
SCHEMBL7982605 0.83 MEN1 (0.76) MEN1CYP3A4CYP2D6CYP2C9KMT2A
SCHEMBL7995942 0.82 OPRL1 (0.75) MEN1CYP3A4CYP2D6CYP2C9KMT2A
SCHEMBL7760221 0.82 MEN1 (0.75) MEN1CYP3A4CYP2D6CYP2C9KMT2A
SCHEMBL20187136 0.82 MEN1 (0.66) MEN1CYP3A4CYP2D6CYP2C9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6277991-B1 FOR TREATMENT OF MIGRAINE, NON-INSULIN DEPENDENT DIABETES MELLITUS, SEPSIS, INFLAMMATION, INCONTINENCE, VASOMOTOR DISTURBANCES SUCH AS HOT FLUSHES OR HOT FLASHES NOVO NORDISK A/S (DK) 2001-08-21 US disclosed