SCHEMBL7994718

SCHEMBL7994718

COc1ccc2c(C)cc(-c3nc(C(F)(F)F)cs3)nc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.40
ALDH1A1 P00352 6/20 0.40
HPGD P15428 3/20 0.40
TSHR P16473 1/20 0.40
HBB P68871 1/20 0.40
HSD17B10 Q99714 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C19 P33261 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MAPT P10636 6/20 0.40
NPSR1 Q6W5P4 2/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
CYP1A1 P04798 2/20 0.38
CYP1B1 Q16678 2/20 0.38
ACHE P22303 1/20 0.38
LMNA P02545 1/20 0.37
NT5E P21589 1/20 0.37
PRNP P04156 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8003565 0.87 KDM4E (0.41) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL7993555 0.80 PDE3B (0.39) KDM4EALDH1A1HPGDHSD17B10CYP1A2
SCHEMBL7993028 0.80 KDM4E (0.38) KDM4EALDH1A1HPGDTSHRHSD17B10
SCHEMBL12362342 0.80 KDM4E (0.41) KDM4EALDH1A1HPGDTSHRHBB
SCHEMBL8005279 0.80 MEN1 (0.36) KDM4EALDH1A1CYP1A2MEN1KMT2A
SCHEMBL8006158 0.79 IGF1R (0.35) MEN1KMT2AMAPTNPC1PTGS1
SCHEMBL577700 0.78 KMT2A (0.40) KDM4EALDH1A1HPGDL3MBTL1CYP1A2
SCHEMBL8006684 0.77 NPC1 (0.37) KDM4EALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL7996053 0.76 KDM4E (0.36) KDM4EALDH1A1L3MBTL1MAPTNPSR1
SCHEMBL11904911 0.75 CYP1B1 (0.40) KDM4EALDH1A1HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed