SCHEMBL7996053

SCHEMBL7996053

COc1ccc2c(C)cc(-c3nc(C(F)(F)F)cs3)nc2c1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
RAB9A P51151 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PDE4B Q07343 10/20 0.35
PDE4A P27815 5/20 0.35
PDE4C Q08493 5/20 0.35
PDE4D Q08499 5/20 0.35
PDE11A Q9HCR9 1/20 0.35
CYP19A1 P11511 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
PTGES O14684 1/20 0.34
RORC P51449 1/20 0.34
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3674311 0.90 PDE4B (0.37) KDM4EMAPTNPC1LMNARAB9A
SCHEMBL7993028 0.89 KDM4E (0.38) KDM4EMAPTNPC1LMNARAB9A
SCHEMBL8003756 0.88 KDM4E (0.36) KDM4EMAPTNPC1LMNARAB9A
SCHEMBL313131 0.88 PDE4B (0.36) MAPTRAB9APDE4BPDE4APDE4C
SCHEMBL8006684 0.88 NPC1 (0.37) KDM4EMAPTNPC1LMNARAB9A
SCHEMBL13090548 0.85 MAPT (0.40) KDM4EMAPTNPC1LMNARAB9A
SCHEMBL8005665 0.82 RORC (0.37) KDM4EMAPTNPC1LMNARAB9A
SCHEMBL8006049 0.80 MAPT (0.36) KDM4EMAPTNPC1LMNARAB9A
SCHEMBL8005668 0.79 C1S (0.36) KDM4EMAPTNPC1LMNARAB9A
SCHEMBL8006158 0.79 IGF1R (0.35) MAPTNPC1PTGESPTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed