SCHEMBL8003565

SCHEMBL8003565

COc1ccc2c(N)cc(-c3nc(C(F)(F)F)cs3)nc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ACHE P22303 2/20 0.39
ALDH1A1 P00352 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
APP P05067 1/20 0.38
CYP1A1 P04798 3/20 0.37
CYP1B1 Q16678 3/20 0.37
ABCC8 Q09428 1/20 0.37
KCNJ11 Q14654 1/20 0.37
NT5E P21589 1/20 0.36
PLK4 O00444 1/20 0.35
DYRK3 O43781 1/20 0.35
MAP4K4 O95819 1/20 0.35
CDK1 P06493 1/20 0.35
RET P07949 1/20 0.35
ROS1 P08922 1/20 0.35
FGFR1 P11362 1/20 0.35
FER P16591 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7994718 0.87 KDM4E (0.40) KDM4EMEN1KMT2AACHEALDH1A1
SCHEMBL8005879 0.81 KDM4E (0.42) KDM4EMEN1KMT2AACHEALDH1A1
SCHEMBL15216084 0.80 ACHE (0.40) KDM4EMEN1KMT2AACHEALDH1A1
SCHEMBL8005887 0.80 SLC2A1 (0.40) KDM4EALDH1A1SMN1; SMN2KDRNPC1
SCHEMBL15216086 0.80 PDE4B (0.35) KDM4EMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL15216081 0.78 KDM4E (0.35) KDM4EMEN1KMT2AACHEALDH1A1
SCHEMBL7996051 0.77 KMT2A (0.37) KDM4EMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL577700 0.77 KMT2A (0.40) KDM4EMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL8003756 0.76 KDM4E (0.36) KDM4EMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL7996056 0.76 SLC2A1 (0.35) KDM4EMEN1KMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250174-B1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS INC (US) 2013-08-28 EP disclosed
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed