SCHEMBL7995572

SCHEMBL7995572

CN(C)c1ccc(-c2nc(C(=O)Nc3nccs3)c(-c3ccc(C(F)(F)F)cc3)[nH]2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 5/20 0.47
GCK P35557 1/20 0.44
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
AURKB Q96GD4 1/20 0.43
AURKC Q9UQB9 1/20 0.43
MAPT P10636 4/20 0.42
TP53 P04637 1/20 0.42
MAPK1 P28482 3/20 0.41
TSHR P16473 2/20 0.41
POLB P06746 1/20 0.41
RAB9A P51151 1/20 0.41
MEN1 O00255 5/20 0.41
KMT2A Q03164 5/20 0.41
GAA P10253 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
ALDH1A1 P00352 3/20 0.41
HPGD P15428 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7992218 0.91 AURKA (0.47) AURKACYP3A4CYP2D6CYP2C9AURKB
SCHEMBL7988697 0.90 GCK (0.42) AURKAGCKMAPTMAPK1TSHR
SCHEMBL7978582 0.90 RAB9A (0.52) GCKMAPTMAPK1TSHRPOLB
SCHEMBL7991779 0.90 AURKA (0.49) AURKACYP3A4CYP2D6CYP2C9AURKB
SCHEMBL7977577 0.89 RAB9A (0.47) GCKMAPTTP53MAPK1TSHR
SCHEMBL7991866 0.89 MAPK1 (0.51) GCKMAPTMAPK1TSHRPOLB
SCHEMBL7989403 0.89 AURKA (0.51) AURKACYP3A4CYP2D6CYP2C9AURKB
SCHEMBL7977619 0.88 RAB9A (0.52) GCKMAPTMAPK1TSHRPOLB
SCHEMBL7992090 0.88 MEN1 (0.52) GCKMAPTMAPK1TSHRPOLB
SCHEMBL7991819 0.88 MEN1 (0.52) AURKAGCKCYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288061-B1 INTERLEUKIN INHIBITORS; ASTHMA, BRONCHODILATOR AGENTS, ANTIALLERGENS WELFIDE CORPORATION (JP) 2001-09-11 US disclosed