SCHEMBL7996473

SCHEMBL7996473

N#CCCCOc1ccc(Cc2[c]ccc(-n3nc(-c4cccnc4)nc3C#N)c2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP11B1 P15538 4/20 0.36
CYP11B2 P19099 4/20 0.36
LTA4H P09960 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
GBA1 P04062 2/20 0.34
CYP19A1 P11511 2/20 0.33
HIF1A Q16665 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
CHRNB2 P17787 2/20 0.33
CHRNA5 P30532 2/20 0.33
CHRNA4 P43681 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7635766 0.79 CACNA1B (0.41) USP2ALDH1A1SMN1; SMN2MAPTHTT
SCHEMBL7635971 0.75 MAPT (0.46) CYP11B1CYP11B2SMN1; SMN2NPC1MAPT
SCHEMBL7996172 0.75 CYP11B1 (0.34) CYP11B1CYP11B2CYP19A1CHRNB2CHRNA5
SCHEMBL8002213 0.73 CYP11B1 (0.37) USP2ALDH1A1CYP11B1CYP11B2SMN1; SMN2
SCHEMBL7630028 0.71 ABCB1 (0.36) ALDH1A1MAPTHTTCYP3A4CYP2D6
SCHEMBL7630588 0.68 TSHR (0.42) ALDH1A1SMN1; SMN2NPC1MAPTHTT
SCHEMBL7238638 0.66 CACNA1B (0.41) USP2ALDH1A1SMN1; SMN2HTTCYP19A1
SCHEMBL7631313 0.65 MAPT (0.45) CYP11B1CYP11B2SMN1; SMN2NPC1MAPT
SCHEMBL7233535 0.65 CACNA1B (0.42) ALDH1A1MAPTCYP3A4CYP2D6CYP2C9
SCHEMBL7239115 0.63 MAPT (0.46) CYP11B1CYP11B2SMN1; SMN2NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001072740-A1 SUBSTITUTED 1-(4-AMINOPHENYL) TRIAZOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-10-04 WO claimed