SCHEMBL7997651

SCHEMBL7997651

N#Cc1ccccc1N1CCC(N2CC(N)C2)CC1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 2/20 0.43
CD274 Q9NZQ7 2/20 0.43
C5AR1 P21730 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GRM5 P41594 1/20 0.40
TRPC6 Q9Y210 3/20 0.39
CYP3A4 P08684 1/20 0.39
TRPC3 Q13507 1/20 0.39
DPP4 P27487 5/20 0.39
AR P10275 1/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
MBTD1 Q05BQ5 1/20 0.37
L3MBTL3 Q96JM7 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CHRM4 P08173 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7843992 0.93 PDCD1 (0.42) PDCD1CD274C5AR1KDM4EALDH1A1
SCHEMBL8005731 0.85 C5AR1 (0.41) PDCD1CD274C5AR1KDM4EALDH1A1
SCHEMBL2261269 0.84 KDM4E (0.47) C5AR1KDM4EALDH1A1GRM5CYP3A4
SCHEMBL8005728 0.83 GAA (0.53) PDCD1CD274C5AR1KDM4EGRM5
SCHEMBL12835705 0.83 DPP4 (0.47) KDM4EALDH1A1GRM5DPP4
SCHEMBL20129683 0.83 DPP4 (0.47) KDM4EALDH1A1GRM5DPP4
Hydrochloric Acid SCHEMBL1514528 0.81 DPP4 (0.47) KDM4EALDH1A1GRM5DPP4
Hydrochloric Acid SCHEMBL1514285 0.81 DPP4 (0.47) KDM4EALDH1A1GRM5DPP4
SCHEMBL20129652 0.81 GRM1 (0.46) KDM4EALDH1A1GRM5DPP4AR
SCHEMBL8008071 0.80 CHRM4 (0.41) PDCD1CD274C5AR1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143750-A NITROGEN HETEROCYCLIC COMPOUNDS AS ENZYME INHIBITORS, FOR PROSTATE PROBLEMS AND MUSCLE RELAXANTS MERCK & CO., INC. (US) 2000-11-07 US disclosed