SCHEMBL8008071

SCHEMBL8008071

N#Cc1ccccc1N1CCC(N2CCC(CN)C2)CC1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 1/20 0.41
C5AR1 P21730 1/20 0.40
PDCD1 Q15116 2/20 0.39
CD274 Q9NZQ7 2/20 0.39
BPTF Q12830 1/20 0.39
DRD4 P21917 2/20 0.37
DRD2 P14416 1/20 0.37
GRM5 P41594 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GRM2 Q14416 1/20 0.37
CYP3A4 P08684 1/20 0.36
CHRM1 P11229 1/20 0.35
KDM1A O60341 1/20 0.35
HTR7 P34969 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8008422 0.93 PDCD1 (0.43) CHRM4C5AR1PDCD1CD274
SCHEMBL8007983 0.92 PDCD1 (0.43) CHRM4C5AR1PDCD1CD274DRD4
SCHEMBL8005731 0.92 C5AR1 (0.41) CHRM4C5AR1PDCD1CD274DRD4
SCHEMBL8214004 0.86 BPTF (0.47) CHRM4C5AR1BPTFDRD4DRD2
SCHEMBL8222584 0.86 CHRM4 (0.46) CHRM4C5AR1DRD4DRD2GRM5
SCHEMBL30163903 0.86 CHRM4 (0.46) CHRM4C5AR1DRD4DRD2GRM5
SCHEMBL7843992 0.84 PDCD1 (0.42) C5AR1PDCD1CD274DRD4DRD2
Trifluoroacetic Acid SCHEMBL7996067 0.83 CHRM4 (0.42) CHRM4C5AR1DRD4DRD2KDM4E
SCHEMBL8006055 0.80 PDCD1 (0.43) CHRM4C5AR1PDCD1CD274
SCHEMBL7997651 0.80 PDCD1 (0.43) CHRM4C5AR1PDCD1CD274DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143750-A NITROGEN HETEROCYCLIC COMPOUNDS AS ENZYME INHIBITORS, FOR PROSTATE PROBLEMS AND MUSCLE RELAXANTS MERCK & CO., INC. (US) 2000-11-07 US disclosed