SCHEMBL7998599

SCHEMBL7998599

O=C1OC2(CC2)C(c2ccncc2)=C1c1ccc(CCc2ccc3ccccc3n2)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 8/20 0.42
WNT3A P56704 1/20 0.38
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
NPC1 O15118 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
AR P10275 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
RAB9A P51151 1/20 0.35
CYSLTR2 Q9NS75 1/20 0.34
CYSLTR1 Q9Y271 1/20 0.34
ALOX5 P09917 1/20 0.34
FFAR1 O14842 1/20 0.33
AKR1B1 P15121 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1419874 0.84 PDE10A (0.56) PDE10ACYSLTR2CYSLTR1
SCHEMBL8003087 0.75 CYSLTR1 (0.35) PDE10ACYSLTR2CYSLTR1ALOX5FFAR1
SCHEMBL3328917 0.74 PDE10A (0.56) PDE10ACYSLTR2CYSLTR1ALOX5
SCHEMBL1420246 0.71 PDE10A (0.56) PDE10ACYSLTR2CYSLTR1
SCHEMBL30123334 0.67 MAPK8 (0.57) PDE10A
SCHEMBL3269253 0.67 MAPK8 (0.57) PDE10A
SCHEMBL1419880 0.67 GPBAR1 (0.52) PDE10ACYSLTR2CYSLTR1ALOX5FFAR1
SCHEMBL12169148 0.67 PDE10A (0.52) PDE10ACYSLTR2CYSLTR1ALOX5
SCHEMBL3329402 0.66 PDE10A (0.53) PDE10ACYSLTR2CYSLTR1
SCHEMBL8007284 0.66 FFAR1 (0.38) PDE10ACYP1A2CYSLTR2CYSLTR1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009158393-A1 1, 2 DISUBSTITUTED HETEROCYCLIC COMPOUNDS ENVIVO PHARMACEUTICALS, INC. (US) 2009-12-30 WO disclosed