SCHEMBL8000212

SCHEMBL8000212

NC(=C1CC1)c1nc2ccccc2nc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.50
ALDH1A1 P00352 4/20 0.50
KDM4E B2RXH2 3/20 0.50
GAA P10253 2/20 0.50
HPGD P15428 2/20 0.50
HSD17B10 Q99714 2/20 0.50
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
NUDT1 P36639 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
IKBKB O14920 1/20 0.39
HRH3 Q9Y5N1 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NPC1 O15118 1/20 0.36
USP2 O75604 1/20 0.36
POLB P06746 1/20 0.36
CACNA1B Q00975 1/20 0.36
APBA1 Q02410 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4101721 0.75 ALDH1A1 (0.56) MAPTALDH1A1KDM4EGAAHPGD
SCHEMBL12629768 0.72 MAPT (0.52) MAPTALDH1A1KDM4EGAAHPGD
SCHEMBL1759326 0.71 ALDH1A1 (0.72) MAPTALDH1A1KDM4EGAAHPGD
SCHEMBL29444102 0.70 MAPT (1.00) MAPTALDH1A1KDM4EGAAHPGD
SCHEMBL503252 0.70 MAPT (1.00) MAPTALDH1A1KDM4EGAAHPGD
SCHEMBL15722184 0.69 MAPT (0.54) MAPTALDH1A1KDM4EGAAHPGD
SCHEMBL12630186 0.69 MAPT (0.54) MAPTALDH1A1KDM4EGAAHPGD
SCHEMBL7990357 0.69 MAPT (0.54) MAPTALDH1A1KDM4EGAAHPGD
SCHEMBL12630110 0.67 MAPT (0.50) MAPTALDH1A1KDM4EGAAHPGD
SCHEMBL12663994 0.66 MAPT (0.48) MAPTALDH1A1KDM4EGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111442-A1 AMINO-QUINOXALINE AND AMINO-QUINOLINE COMPOUNDS FOR USE AS ADENOSINE A2a RECEPTOR ANTAGONISTS SCHERING CORPORATION (US) 2009-09-11 WO disclosed