SCHEMBL8001013

SCHEMBL8001013

Fc1cccc2c1C(CNC1CC1)CN2Cc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 4/20 0.48
CACNA1H O95180 4/20 0.48
CACNA1I Q9P0X4 4/20 0.48
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
BRD4 O60885 2/20 0.39
BCHE P06276 6/20 0.38
ACHE P22303 6/20 0.38
BACE1 P56817 6/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SIGMAR1 Q99720 1/20 0.37
MTNR1A P48039 2/20 0.37
MTNR1B P49286 2/20 0.37
SIRT1 Q96EB6 1/20 0.36
ALOX12 P18054 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7999586 0.86 BRD4 (0.39) CACNA1GCACNA1HCACNA1IBRD4BCHE
SCHEMBL8002826 0.77 BCHE (0.44) CACNA1GCACNA1HCACNA1IBCHEACHE
SCHEMBL13625710 0.72 BCHE (0.43) CACNA1GCACNA1HCACNA1IBRD4BCHE
SCHEMBL7992727 0.71 BRD4 (0.50) CACNA1GCACNA1HCACNA1IKDM4EBRD4
SCHEMBL7990909 0.64 OPRL1 (0.35)
SCHEMBL9437321 0.62 ACHE (0.60) BCHEACHEBACE1
SCHEMBL28305302 0.62 KDM4E (0.58) KDM4EGAABCHEACHEBACE1
SCHEMBL28169202 0.62 CXCR4 (0.68) BCHEACHEBACE1SIGMAR1
SCHEMBL1518407 0.61 ACHE (0.47) BCHEACHEBACE1SIGMAR1
SCHEMBL7999624 0.61 LIPG (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009140769-A1 3, 4 - SUBSTITUTED PIPERIDINE DERIVATIVES AS RENIN INHIBITORS MERCK FROSST CANADA LTD. (CA) 2009-11-26 WO disclosed