SCHEMBL8002279

SCHEMBL8002279

COc1ccc2c(O[C@H]3C[C@@H](C(=O)O)N(C(=O)OC(C)(C)C)C3)cc(-c3nc(C(F)(F)F)cs3)nc2c1Cl

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
UCHL1 P09936 1/20 0.38
ABCC1 P33527 1/20 0.35
ABCC2 Q92887 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35
CTSB P07858 1/20 0.35
PPP3CB P16298 1/20 0.35
PDE4B Q07343 3/20 0.33
PDE11A Q9HCR9 1/20 0.33
PDE10A Q9Y233 1/20 0.33
P2RX3 P56373 2/20 0.32
RORC P51449 2/20 0.32
MCL1 Q07820 5/20 0.32
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32
BCL2 P10415 1/20 0.31
BCL2L1 Q07817 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL313037 0.92 UCHL1 (0.39) UCHL1CTSBPPP3CBPDE4BPDE11A
SCHEMBL3808212 0.92 UCHL1 (0.39) UCHL1CTSBPPP3CBPDE4BPDE11A
SCHEMBL2213932 0.89 UCHL1 (0.38) UCHL1ABCC1ABCC2ABCG2CTSB
SCHEMBL313204 0.89 UCHL1 (0.38) UCHL1ABCC1ABCC2ABCG2CTSB
SCHEMBL1101736 0.89 UCHL1 (0.38) UCHL1ABCC1ABCC2ABCG2CTSB
SCHEMBL8002276 0.88 PDE4B (0.33) UCHL1ABCC1ABCC2ABCG2CTSB
SCHEMBL312718 0.86 UCHL1 (0.37) UCHL1CTSBPPP3CBPDE4BPDE11A
SCHEMBL312719 0.86 UCHL1 (0.37) UCHL1CTSBPPP3CBPDE4BPDE11A
SCHEMBL8002444 0.85 UCHL1 (0.36) UCHL1ABCC1ABCC2ABCG2CTSB
SCHEMBL15216085 0.85 UCHL1 (0.36) UCHL1ABCC1ABCC2ABCG2CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250174-B1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS INC (US) 2013-08-28 EP disclosed
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed