SCHEMBL8002276

SCHEMBL8002276

COOC[C@@H]1C[C@H](Oc2cc(-c3nc(C(F)(F)F)cs3)nc3c(Cl)c(OC)ccc23)CN1C(=O)OC(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 4/20 0.33
PDE11A Q9HCR9 2/20 0.33
PDE10A Q9Y233 2/20 0.33
ABCC1 P33527 1/20 0.32
ABCC2 Q92887 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
CTSB P07858 1/20 0.32
PPP3CB P16298 1/20 0.32
UCHL1 P09936 1/20 0.31
RORC P51449 2/20 0.31
PPARD Q03181 1/20 0.31
PPARA Q07869 1/20 0.31
PDE4A P27815 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8006736 0.93 CTSS (0.33) PDE4BPDE11APDE10ACTSBPPP3CB
SCHEMBL8002279 0.88 UCHL1 (0.38) PDE4BPDE11APDE10AABCC1ABCC2
SCHEMBL10247425 0.82 PIK3CD (0.35) UCHL1
SCHEMBL8002444 0.81 UCHL1 (0.36) ABCC1ABCC2ABCG2CTSBPPP3CB
SCHEMBL15216085 0.81 UCHL1 (0.36) ABCC1ABCC2ABCG2CTSBPPP3CB
SCHEMBL3808212 0.80 UCHL1 (0.39) PDE4BPDE11APDE10ACTSBPPP3CB
SCHEMBL313037 0.80 UCHL1 (0.39) PDE4BPDE11APDE10ACTSBPPP3CB
SCHEMBL312718 0.80 UCHL1 (0.37) PDE4BPDE11APDE10ACTSBPPP3CB
SCHEMBL312719 0.80 UCHL1 (0.37) PDE4BPDE11APDE10ACTSBPPP3CB
SCHEMBL10247252 0.77 PIK3CD (0.35) UCHL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed