SCHEMBL8002464

SCHEMBL8002464

C1=CC2(CCN(CCCCN3CCC4(C=Cc5ccccc5O4)CC3)CC2)Oc2ccccc21

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 2/20 0.66
ADRA1D P25100 1/20 0.66
ADRA1B P35368 1/20 0.66
HTR2C P28335 7/20 0.57
HTR2B P41595 1/20 0.57
DRD2 P14416 3/20 0.51
HTR2A P28223 3/20 0.51
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
SCD O00767 1/20 0.41
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7442602 0.91 ADRA1D (0.60) ADRA1AADRA1DADRA1BHTR2CHTR2B
SCHEMBL3413391 0.83 HTR2C (0.62) ADRA1AADRA1DADRA1BHTR2CHTR2B
SCHEMBL4275257 0.83 HDAC3 (0.58) ADRA1AADRA1DADRA1BHTR2CHTR2B
SCHEMBL7370885 0.80 HTR2C (0.62) ADRA1AADRA1DADRA1BHTR2CHTR2B
Hydrochloric Acid SCHEMBL4269341 0.80 ADRA1D (0.54) ADRA1AADRA1DADRA1BHTR2CHTR2B
SCHEMBL3552550 0.77 HTR2C (0.72) ADRA1AADRA1DADRA1BHTR2CHTR2B
SCHEMBL8010432 0.77 ADRA1D (0.54) ADRA1AADRA1DADRA1BHTR2CHTR2B
SCHEMBL12481728 0.77 HTR2C (0.57) ADRA1AADRA1DADRA1BHTR2CHTR2B
SCHEMBL1115308 0.76 HTR2C (0.70) ADRA1AADRA1DADRA1BHTR2CHTR2B
SCHEMBL3709748 0.74 HTR2C (0.55) ADRA1AADRA1DADRA1BHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0649407-B1 DIMERIC PIPERIDINE, TETRAHYDROPYRIDINE AND PIPERAZINE DERIVATIVES LUNDBECK & CO AS H (DK) 1998-08-05 EP claimed
US-6090808-A PSYCHOLOGICAL DISORDERS; ANTICONVULSANTS H. LUNDBECK A/S (DK) 2000-07-18 US disclosed
EP-0649407-B1 DIMERIC PIPERIDINE, TETRAHYDROPYRIDINE AND PIPERAZINE DERIVATIVES LUNDBECK & CO AS H (DK) 1998-08-05 EP disclosed
US-5658921-A POTENT SIGMA RECEPTOR LIGANDS; WATER SOLUBILITY; SYMMETRY H. LUNDBECK A/S (DK) 1997-08-19 US disclosed