SCHEMBL8002791

SCHEMBL8002791

CCc1nc2c(cnn2CC)c(NC2CCOCC2)c1CNC(=O)NCc1ccc(Cl)c(-c2cccc(CC3CCNCC3)c2)c1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 12/20 0.44
MAPK1 P28482 6/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
KCNH2 Q12809 1/20 0.36
PTGES O14684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13750943 0.96 PDE4B (0.43) PDE4BMAPK1CHRM2CHRM1CHRM3
SCHEMBL4095656 0.94 PDE4B (0.46) PDE4BMAPK1CHRM2CHRM1CHRM3
SCHEMBL8003330 0.93 PDE4B (0.45) PDE4BMAPK1CHRM2CHRM1CHRM3
SCHEMBL3429059 0.93 PDE4B (0.49) PDE4BMAPK1
SCHEMBL8007729 0.93 PDE4B (0.44) PDE4BMAPK1CHRM2CHRM1CHRM3
SCHEMBL8008701 0.93 PDE4B (0.44) PDE4BMAPK1
SCHEMBL8002739 0.92 PDE4B (0.43) PDE4BMAPK1CHRM2CHRM1CHRM3
SCHEMBL8014879 0.91 PDE4B (0.44) PDE4BCHRM2CHRM1CHRM3
SCHEMBL3427552 0.91 PDE4B (0.39) PDE4BMAPK1CHRM2CHRM1CHRM3
SCHEMBL13750940 0.90 PDE4B (0.47) PDE4BMAPK1CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100170-A1 DUAL PHARMACOPHORES - PDE4-MUSCARINIC ANTAGONISTICS GLAXO GROUP LIMITED (GB) 2009-08-13 WO disclosed