SCHEMBL8003330

SCHEMBL8003330

CCc1nc2c(cnn2CC)c(NC2CCOCC2)c1CNC(=O)NCc1ccc(C)c(-c2cccc(CC3CCNCC3)c2)c1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 14/20 0.45
MAPK1 P28482 3/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
KCNH2 Q12809 1/20 0.36
PDE3B Q13370 1/20 0.33
PDE7A Q13946 1/20 0.33
PDE3A Q14432 1/20 0.33
USP28 Q96RU2 1/20 0.33
USP25 Q9UHP3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13750944 0.96 PDE4B (0.43) PDE4BMAPK1CHRM2CHRM1CHRM3
SCHEMBL4099149 0.94 PDE4B (0.46) PDE4BMAPK1CHRM2CHRM1CHRM3
SCHEMBL3429059 0.94 PDE4B (0.49) PDE4BMAPK1PDE7A
SCHEMBL8007729 0.93 PDE4B (0.44) PDE4BMAPK1CHRM2CHRM1CHRM3
SCHEMBL8002791 0.93 PDE4B (0.44) PDE4BMAPK1CHRM2CHRM1CHRM3
SCHEMBL8011054 0.93 PDE4B (0.45) PDE4BMAPK1
SCHEMBL8002739 0.92 PDE4B (0.43) PDE4BMAPK1CHRM2CHRM1CHRM3
SCHEMBL13750940 0.90 PDE4B (0.47) PDE4BMAPK1CHRM2CHRM1CHRM3
SCHEMBL3426907 0.90 PDE4B (0.41) PDE4BMAPK1CHRM2CHRM1CHRM3
SCHEMBL13750943 0.89 PDE4B (0.43) PDE4BMAPK1CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100170-A1 DUAL PHARMACOPHORES - PDE4-MUSCARINIC ANTAGONISTICS GLAXO GROUP LIMITED (GB) 2009-08-13 WO disclosed