SCHEMBL8007729

SCHEMBL8007729

CCc1nc2c(cnn2CC)c(NC2CCOCC2)c1CNC(=O)NCc1ccc(F)c(-c2cccc(CC3CCNCC3)c2)c1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 12/20 0.44
CHRM3 P20309 6/20 0.44
CHRM2 P08172 2/20 0.44
CHRM1 P11229 2/20 0.44
KCNH2 Q12809 1/20 0.44
MAPK1 P28482 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13750942 0.96 PDE4B (0.43) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL4095093 0.94 PDE4B (0.46) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL1364219 0.94 CHRM3 (0.51) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL8003330 0.93 PDE4B (0.45) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL3429059 0.93 PDE4B (0.49) PDE4BMAPK1
SCHEMBL8002791 0.93 PDE4B (0.44) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL8014793 0.93 PDE4B (0.44) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL8002739 0.92 PDE4B (0.43) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL3428370 0.90 PDE4B (0.40) PDE4BCHRM3CHRM2CHRM1KCNH2
SCHEMBL13750940 0.90 PDE4B (0.47) PDE4BCHRM3CHRM2CHRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100170-A1 DUAL PHARMACOPHORES - PDE4-MUSCARINIC ANTAGONISTICS GLAXO GROUP LIMITED (GB) 2009-08-13 WO disclosed