SCHEMBL8006436

SCHEMBL8006436

CCCc1c(OCCCNc2ccc(CC(=O)OC)cc2Cl)ccc2c(C(F)(F)F)noc12

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 20/20 0.69
NR1H2 P55055 18/20 0.69
PPARD Q03181 14/20 0.69
PPARA Q07869 11/20 0.69
PPARG P37231 8/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7040305 0.93 NR1H3 (0.81) NR1H3NR1H2PPARDPPARAPPARG
SCHEMBL7044849 0.88 PPARD (0.54) NR1H3NR1H2PPARDPPARAPPARG
SCHEMBL14465277 0.87 NR1H3 (0.62) NR1H3NR1H2PPARDPPARAPPARG
SCHEMBL7044517 0.85 PPARD (0.86) NR1H3NR1H2PPARDPPARAPPARG
SCHEMBL7046590 0.85 NR1H3 (0.69) NR1H3NR1H2PPARDPPARAPPARG
SCHEMBL5203759 0.83 PPARD (0.83) NR1H3NR1H2PPARDPPARAPPARG
SCHEMBL14465348 0.83 NR1H2 (0.57) NR1H3NR1H2PPARDPPARAPPARG
SCHEMBL7039181 0.81 PPARD (0.62) NR1H3NR1H2PPARDPPARAPPARG
SCHEMBL7046131 0.81 PPARG (0.73) NR1H3NR1H2PPARDPPARAPPARG
SCHEMBL7042314 0.80 NR1H3 (0.72) NR1H3NR1H2PPARDPPARAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090836-A DIETETICS; ADJUSTMENT OF TRIGLYCERIDE CONCENTRATION MERCK & CO., INC. (US) 2000-07-18 US disclosed
EP-0882029-A1 HETEROCYCLIC DERIVATIVES AS ANTIDIABETIC AND ANTIOBESITY AGENTS Merck & Co., Inc. (US) 1998-12-09 EP disclosed
WO-1997028137-A1 HETEROCYCLIC DERIVATIVES AS ANTIDIABETIC AND ANTIOBESITY AGENTS MERCK & CO., INC. (US) 1997-08-07 WO disclosed