SCHEMBL8006887

SCHEMBL8006887

COc1ccc2c(N)nc(-c3nc(C(C)C)cs3)nc2c1Cl

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.36
ADORA1 P30542 3/20 0.36
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
APLNR P35414 1/20 0.33
ILK Q13418 1/20 0.32
PDPK1 O15530 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
RAD52 P43351 1/20 0.31
CYP19A1 P11511 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL313190 0.87 APLNR (0.33) ALDH1A1KDM4EAPLNRTDP1CYP19A1
SCHEMBL8004421 0.87 ADORA2A (0.39) ADORA2AADORA1ALDH1A1KDM4EAPLNR
SCHEMBL8003752 0.86 ADORA2A (0.38) ADORA2AADORA1ALDH1A1APLNRRAD52
SCHEMBL8006162 0.81 ALDH1A1 (0.37) ALDH1A1KDM4EAPLNRTDP1HTR2A
SCHEMBL10272030 0.79 ALDH1A1 (0.34) ALDH1A1KDM4EAPLNRTDP1CYP19A1
SCHEMBL1496428 0.78 APLNR (0.35) ALDH1A1KDM4EAPLNRPDPK1TDP1
SCHEMBL996629 0.78 ALDH1A1 (0.33) ALDH1A1KDM4EAPLNRTDP1CYP19A1
SCHEMBL577814 0.77 ALDH1A1 (0.33) ALDH1A1KDM4EAPLNRTDP1CYP19A1
SCHEMBL8003339 0.77 POLB (0.39) ADORA2AADORA1ALDH1A1KDM4ERAD52
SCHEMBL995496 0.76 ALDH1A1 (0.35) ALDH1A1KDM4EAPLNRTDP1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed