SCHEMBL8007932

SCHEMBL8007932

COc1ccc2c(N)cc(-c3csc(C(C)C)n3)nc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
ACHE P22303 1/20 0.38
CYP3A4 P08684 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
MEN1 O00255 1/20 0.38
GFER P55789 1/20 0.38
KMT2A Q03164 1/20 0.38
GAA P10253 1/20 0.37
APP P05067 1/20 0.36
CYP1A1 P04798 1/20 0.36
CYP1B1 Q16678 1/20 0.36
SLC2A1 P11166 1/20 0.36
MPO P05164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15216113 0.86 KDM4E (0.42) ALDH1A1SMN1; SMN2KDM4EPOLBMAPT
SCHEMBL15216084 0.80 ACHE (0.40) ALDH1A1SMN1; SMN2KDM4ENPC1POLB
SCHEMBL7993475 0.80 PDE3B (0.37) ALDH1A1SMN1; SMN2KDM4ENPC1POLB
SCHEMBL15216087 0.79 SLC2A1 (0.42) ALDH1A1SMN1; SMN2KDM4ENPC1GAA
SCHEMBL8011476 0.79 MEN1 (0.36) ALDH1A1SMN1; SMN2KDM4ENPC1POLB
SCHEMBL8006881 0.77 MEN1 (0.35) ALDH1A1SMN1; SMN2KDM4ENPC1POLB
SCHEMBL8008296 0.77 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2KDM4ENPC1POLB
SCHEMBL577492 0.76 SMN1; SMN2 (0.36) ALDH1A1SMN1; SMN2KDM4ENPC1POLB
SCHEMBL8008865 0.75 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2KDM4ENPC1POLB
SCHEMBL8008888 0.75 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2KDM4ENPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250174-B1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS INC (US) 2013-08-28 EP disclosed
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed