SCHEMBL8007983

SCHEMBL8007983

N#Cc1ccccc1N1CCC(N2CCC(CN)CC2)CC1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 2/20 0.43
CD274 Q9NZQ7 2/20 0.43
CHRM4 P08173 1/20 0.42
C5AR1 P21730 1/20 0.41
CHRM1 P11229 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
DRD2 P14416 2/20 0.38
DRD4 P21917 2/20 0.38
GRM5 P41594 1/20 0.38
MBTD1 Q05BQ5 1/20 0.38
L3MBTL3 Q96JM7 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ADRA1D P25100 1/20 0.37
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
CYP3A4 P08684 1/20 0.37
CXCR4 P61073 1/20 0.37
GRIN2B Q13224 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8008071 0.92 CHRM4 (0.41) PDCD1CD274CHRM4C5AR1CHRM1
SCHEMBL30163903 0.92 CHRM4 (0.46) CHRM4C5AR1KDM4EALDH1A1DRD2
SCHEMBL8222584 0.92 CHRM4 (0.46) CHRM4C5AR1KDM4EALDH1A1DRD2
SCHEMBL8005731 0.89 C5AR1 (0.41) PDCD1CD274CHRM4C5AR1KDM4E
SCHEMBL8008422 0.85 PDCD1 (0.43) PDCD1CD274CHRM4C5AR1MBTD1
SCHEMBL8214004 0.83 BPTF (0.47) CHRM4C5AR1KDM4EALDH1A1DRD2
SCHEMBL7843992 0.81 PDCD1 (0.42) PDCD1CD274C5AR1KDM4EALDH1A1
SCHEMBL8007979 0.79 GAA (0.58) PDCD1CD274CHRM4CHRM1KDM4E
SCHEMBL7997651 0.79 PDCD1 (0.43) PDCD1CD274CHRM4C5AR1KDM4E
SCHEMBL30626544 0.79 PDCD1 (0.46) PDCD1CD274C5AR1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143750-A NITROGEN HETEROCYCLIC COMPOUNDS AS ENZYME INHIBITORS, FOR PROSTATE PROBLEMS AND MUSCLE RELAXANTS MERCK & CO., INC. (US) 2000-11-07 US disclosed