SCHEMBL8008068

SCHEMBL8008068

N#Cc1ccccc1N1CCC(N2CCC(C(N)=O)C2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.54
KDM4E B2RXH2 1/20 0.53
RECQL P46063 1/20 0.53
AOC3 Q16853 1/20 0.45
CHRM4 P08173 1/20 0.44
GRM5 P41594 1/20 0.44
KDM2B Q8NHM5 2/20 0.42
TSHR P16473 2/20 0.41
SIRT2 Q8IXJ6 1/20 0.41
SIRT1 Q96EB6 1/20 0.41
ALDH1A1 P00352 1/20 0.41
OPRM1 P35372 2/20 0.41
OPRK1 P41145 2/20 0.41
OGFRL1 Q5TC84 2/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
AR P10275 1/20 0.40
NOTUM Q6P988 1/20 0.40
GRM1 Q13255 2/20 0.40
OPRD1 P41143 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8007979 0.94 GAA (0.58) GAAKDM4ERECQLAOC3CHRM4
SCHEMBL8008419 0.93 KDM2B (0.50) GAAKDM4ERECQLCHRM4GRM5
SCHEMBL8005728 0.92 GAA (0.53) GAAKDM4ERECQLAOC3CHRM4
SCHEMBL30332131 0.88 GAA (0.67) GAAKDM4ERECQLCHRM4GRM5
Trifluoroacetic Acid SCHEMBL8006053 0.86 GAA (0.51) GAAKDM4ERECQLAOC3CHRM4
Trifluoroacetic Acid SCHEMBL7996066 0.86 KDM2B (0.45) GAAKDM4ERECQLCHRM4KDM2B
SCHEMBL7843992 0.83 PDCD1 (0.42) GAAKDM4EGRM5ALDH1A1OPRM1
SCHEMBL8006273 0.79 GRM5 (0.46) GAAKDM4ERECQLCHRM4GRM5
SCHEMBL7997651 0.79 PDCD1 (0.43) KDM4ECHRM4GRM5ALDH1A1DRD2
SCHEMBL8008071 0.79 CHRM4 (0.41) KDM4ECHRM4GRM5ALDH1A1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143750-A NITROGEN HETEROCYCLIC COMPOUNDS AS ENZYME INHIBITORS, FOR PROSTATE PROBLEMS AND MUSCLE RELAXANTS MERCK & CO., INC. (US) 2000-11-07 US disclosed